Drug reference

tirzepatide

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Endocrine (Miscellaneous(Hormones))

Mechanism of action

GIP is an incretin hormone that induces insulin secretion in response to a meal (primarily by hyperosmolarity of glucose in the duodenum) to facilitate the metabolism of carbohydrates, fats, and proteins GLP-1 receptor agonists increase insulin secretion in the presence of elevated blood glucose, suppress glucagon postprandially, delay gastric emptying to decrease postprandial glucose

Common side effects

  • Dyspepsia
  • Constipation
  • Decreased appetite
  • Vomiting
  • Nausea
  • Injection site reacation
  • Diarrhea

Related conditions

Frequently asked questions

What drug class is tirzepatide?

tirzepatide belongs to: Endocrine.

How does tirzepatide work?

GIP is an incretin hormone that induces insulin secretion in response to a meal (primarily by hyperosmolarity of glucose in the duodenum) to facilitate the metabolism of carbohydrates, fats, and proteins GLP-1 receptor agonists increase insulin secretion in the presence of elevated blood glucose, suppress glucagon postprandially, delay gastric emptying to decrease postprandial glucose

What are the common side effects of tirzepatide?

Dyspepsia, Constipation, Decreased appetite, Vomiting, Nausea, Injection site reacation, Diarrhea

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