Drug reference

atosiban

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Endocrine (Pituitary Hormones)

Mechanism of action

Atosiban is a synthetic peptide which acts as a competitive antagonist of oxytocin at human uterine oxytocin receptors. Oxytocin causes uterine contractions through a direct effect on membrane bound receptors in the uterus by increasing the concentration of intracellular calcium in the myometrial cells.

Common side effects

  • Pruritus
  • Dizziness
  • Vomiting
  • Headache
  • Nausea
  • Hyperglycaemia
  • Tachycardia

Related conditions

Frequently asked questions

What drug class is atosiban?

atosiban belongs to: Endocrine.

How does atosiban work?

Atosiban is a synthetic peptide which acts as a competitive antagonist of oxytocin at human uterine oxytocin receptors. Oxytocin causes uterine contractions through a direct effect on membrane bound receptors in the uterus by increasing the concentration of intracellular calcium in the myometrial cells.

What are the common side effects of atosiban?

Pruritus, Dizziness, Vomiting, Headache, Nausea, Hyperglycaemia, Tachycardia

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