Drug reference

cycloserine

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Anti Bacterial (Non Beta-Lactams)

Mechanism of action

Cycloserine works as an antibiotic by inhibiting cell-wall biosynthesis in bacteria. As a cyclic analogue of D-alanine, cycloserine acts against two crucial enzymes important in the cytosolic stages of peptidoglycan synthesis: alanine racemase (Alr) and D-alanine:D-alanine ligase (Ddl).

Common side effects

  • Restlessness
  • Drowsiness
  • Confusion
  • Vertigo
  • Cardiac arrhythmia

Contraindications

  • Hypersensitivity Alcohol use Renal dysfunction, severe History of seizure disorder, mental depression, severe anxiety or psychosis

Related conditions

Frequently asked questions

What drug class is cycloserine?

cycloserine belongs to: Anti Bacterial.

How does cycloserine work?

Cycloserine works as an antibiotic by inhibiting cell-wall biosynthesis in bacteria. As a cyclic analogue of D-alanine, cycloserine acts against two crucial enzymes important in the cytosolic stages of peptidoglycan synthesis: alanine racemase (Alr) and D-alanine:D-alanine ligase (Ddl).

What are the common side effects of cycloserine?

Restlessness, Drowsiness, Confusion, Vertigo, Cardiac arrhythmia

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