Drug reference

tolterodine

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Genitourinary (Antimuscarinic)

Mechanism of action

Competitive muscarinic receptor antagonist; decreases bladder contractions; is more specific for bladder than oxybutynin.

Common side effects

  • Dyspepsia
  • Dry mouth
  • Constipation
  • Dizziness
  • Blurred vision

Contraindications

  • Urinary or gastric retention Uncontrolled narrow-angle glaucoma Hypersensitivity to drug or ingredients or to fesoterodine fumarate, which is metabolized to 5-hydroxymethyl tolterodine

Related conditions

Frequently asked questions

What drug class is tolterodine?

tolterodine belongs to: Genitourinary.

How does tolterodine work?

Competitive muscarinic receptor antagonist; decreases bladder contractions; is more specific for bladder than oxybutynin.

What are the common side effects of tolterodine?

Dyspepsia, Dry mouth, Constipation, Dizziness, Blurred vision

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