Riferimento farmaci
Isoconazole
Isoconazole is a medicine in the class anti fungals. It is used for vulvovaginal candidiasis.
- Classe del farmaco: Anti Fungals
- Indicato per: vulvovaginal candidiasis
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In breve
- Classe del farmaco
- Anti Fungals
- Forme farmaceutiche comuni
- crema
- Dosaggi comuni
- 1%, 600 mg, 300 mg
- Nomi commerciali
- 10
- Paesi e mercati
- 3
Per cosa si usa
Come agisce
Azole antifungal agent; inhibits enzyme cytochrome P450 14-alpha-demethylase resulting in ergosterol synthesis inhibition
Dose abituale nell'adulto (sintesi del foglio illustrativo)
600 mg vaginal suppository: Insert 1 suppository qHS x 3 days
Gravidanza e allattamento
- Gravidanza
- Safe Topical and vaginal azole antifungal (e.g. Travogen); little is absorbed. No adequate human data, but topical azoles are not linked to birth defects. Use in the 1st trimester only on medical advice; clotrimazole has the most pregnancy data and is preferred vaginally.
- Allattamento
- Safe Little is absorbed from skin or vagina, so milk levels are expected to be negligible. Topical azoles are considered compatible with breastfeeding. Do not apply to the nipple or breast, and keep the infant's skin away from treated areas.
Effetti indesiderati segnalati
- Irritation
- Allergic contact dermatitis
- Burning
Controindicazioni
- Hypersensitivity to isoconazole or to any of the excipients of the formulation.
Chi deve prestare attenzione
- Avoid contact with the eyes.
- Discontinue treatment if local irritation or a hypersensitivity (sensitisation) reaction develops.
- Some formulations contain cetostearyl alcohol, which may cause local skin reactions such as contact dermatitis.
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- Dosing by age, kidney and liver function, and further dose lines
- Paediatric dosing
- Patient counselling points
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Domande frequenti
What is Isoconazole used for?
Isoconazole is a medicine in the class anti fungals. It is used for Vulvovaginal candidiasis.
What side effects have been reported with Isoconazole?
Irritation, Allergic contact dermatitis, Burning.
Can Isoconazole be taken in pregnancy or while breastfeeding?
Pregnancy: Safe. Topical and vaginal azole antifungal (e.g. Travogen); little is absorbed. No adequate human data, but topical azoles are not linked to birth defects. Use in the 1st trimester only on medical advice; clotrimazole has the most pregnancy data and is preferred vaginally. Breastfeeding: Safe. Little is absorbed from skin or vagina, so milk levels are expected to be negligible. Topical azoles are considered compatible with breastfeeding. Do not apply to the nipple or breast, and keep the infant's skin away from treated areas.
What does Isoconazole interact with?
MediHelp does not list a checked interaction for Isoconazole yet. Always tell your pharmacist about every medicine you take.
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