Drug reference

azilsartan

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Cardiovascular (ARBs)

Mechanism of action

Angiotensin II blocker; displaces angiotensin II from AT1 receptor and may lower blood pressure by antagonizing AT1-induced vasoconstriction, aldosterone release, catecholamine release, arginine vasopressin release, water absorption, and hypertrophic responses

Common side effects

  • Asthenia
  • Fatigue
  • Nausea
  • Musculoskeletal pain
  • Diarrhea

Boxed warnings

  • Discontinue as soon as possible when pregnancy is detected; affects renin-angiotensin system causing oligohydramnios, which may result in fetal injury and/or death

Contraindications

  • Hypersensitivity Do not coadminister with aliskiren in patients with diabetes

Related conditions

Frequently asked questions

What drug class is azilsartan?

azilsartan belongs to: Cardiovascular.

How does azilsartan work?

Angiotensin II blocker; displaces angiotensin II from AT1 receptor and may lower blood pressure by antagonizing AT1-induced vasoconstriction, aldosterone release, catecholamine release, arginine vasopressin release, water absorption, and hypertrophic responses

What are the common side effects of azilsartan?

Asthenia, Fatigue, Nausea, Musculoskeletal pain, Diarrhea

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