Drug reference
cyproterone acetate
For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.
Drug class
Endocrine (Gonadal Hormones)
Mechanism of action
Cyproterone is an antiandrogen. It suppresses the actions of testosterone (and its metabolite dihydrotestosterone) on tissues. It acts by blocking androgen receptors which prevents androgens from binding to them and suppresses luteinizing hormone (which in turn reduces testosterone levels).
Common side effects
- Rash
- Restlessness
- Depressive moods
- Jaundice
- Dyspnoea
Related conditions
Frequently asked questions
What drug class is cyproterone acetate?
cyproterone acetate belongs to: Endocrine.
How does cyproterone acetate work?
Cyproterone is an antiandrogen. It suppresses the actions of testosterone (and its metabolite dihydrotestosterone) on tissues. It acts by blocking androgen receptors which prevents androgens from binding to them and suppresses luteinizing hormone (which in turn reduces testosterone levels).
What are the common side effects of cyproterone acetate?
Rash, Restlessness, Depressive moods, Jaundice, Dyspnoea
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