Drug reference

enzalutamide

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Endocrine (Gonadal Hormones)

Mechanism of action

Androgen receptor inhibitor; competitively inhibits androgen binding to androgen receptors; also inhibits androgen receptor nuclear translocation and interaction with DNA resulting in decreased proliferation and induced cell death

Common side effects

  • Arthralgia
  • Constipation
  • Decreased appetite
  • Back pain
  • Asthenic conditions
  • Hot flush
  • Diarrhea

Related conditions

Frequently asked questions

What drug class is enzalutamide?

enzalutamide belongs to: Endocrine.

How does enzalutamide work?

Androgen receptor inhibitor; competitively inhibits androgen binding to androgen receptors; also inhibits androgen receptor nuclear translocation and interaction with DNA resulting in decreased proliferation and induced cell death

What are the common side effects of enzalutamide?

Arthralgia, Constipation, Decreased appetite, Back pain, Asthenic conditions, Hot flush, Diarrhea

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