Drug reference

fulvestrant

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Endocrine (SERMs)

Mechanism of action

Breast cancer: Competitively binds to estrogen receptors on tumors and other tissue targets, producing nuclear complex that decreases DNA synthesis and inhibits estrogen effects; no estrogen-receptor agonist activity; downregulates estrogen receptors and inhibits breast tumor growth

Common side effects

  • Pharyngitis
  • Asthenia
  • Constipation
  • Nausea
  • Pain
  • Back pain
  • Vasodilatation

Related conditions

Frequently asked questions

What drug class is fulvestrant?

fulvestrant belongs to: Endocrine.

How does fulvestrant work?

Breast cancer: Competitively binds to estrogen receptors on tumors and other tissue targets, producing nuclear complex that decreases DNA synthesis and inhibits estrogen effects; no estrogen-receptor agonist activity; downregulates estrogen receptors and inhibits breast tumor growth

What are the common side effects of fulvestrant?

Pharyngitis, Asthenia, Constipation, Nausea, Pain, Back pain, Vasodilatation

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