Drug reference

letrozole

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Oncology (Aromatase Inhibitors)

Mechanism of action

Aromatase inhibitor - blocks conversion of androgens to estrogens by binding to the heme group of aromatase enzyme, which in turn inhibits its activity

Common side effects

  • Nausea
  • Bone pain
  • Dyspnea
  • Back pain
  • Hot flashes
  • Diaphoresis
  • Night sweats

Related conditions

Frequently asked questions

What drug class is letrozole?

letrozole belongs to: Oncology.

How does letrozole work?

Aromatase inhibitor - blocks conversion of androgens to estrogens by binding to the heme group of aromatase enzyme, which in turn inhibits its activity

What are the common side effects of letrozole?

Nausea, Bone pain, Dyspnea, Back pain, Hot flashes, Diaphoresis, Night sweats

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