Drug interactions
Abemaciclib + Ketoconazole
Severity: Major
Abemaciclib and Ketoconazole: major interaction.
Last updated
For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.
Summary
Ketoconazole markedly raises abemaciclib exposure, increasing the risk of neutropenia, diarrhea, hepatotoxicity and venous thromboembolism.
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Other interactions of Ketoconazole
Other interactions of Abemaciclib
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