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Interazioni tra farmaci

Propranolol + Thioridazine

Gravità: Controindicata

Propranolol and Thioridazine: contraindicated interaction.

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Sintesi

Thioridazine can raise propranolol concentrations, and propranolol can raise thioridazine concentrations. Because thioridazine itself prolongs the QT interval, higher levels increase the risk of torsades de pointes and sudden death.

Cosa significa questa interazione in parole semplici

Propranolol and Thioridazine are not normally used together. Taking them at the same time is expected to cause harm or make one of them unsafe, so a different medicine is usually chosen for one of the two.

Propranolol belongs to Cardiovascular; Thioridazine belongs to Central Nervous System.

Livello di evidenza: Moderate

Perché avviene

Mutual metabolic inhibition involving CYP2D6, with additive cardiac depressant and proarrhythmic effects.

Cosa fare

Avoid concurrent use. If a beta blocker is needed with thioridazine, select one not dependent on CYP2D6 such as atenolol, though thioridazine alternatives are preferred.

Cosa chiedere al farmacista

  • Is there an alternative to one of these two medicines for me?
  • If both are essential, who is monitoring me and how often?
  • Which symptoms mean I should stop and seek help straight away?

Bring a full list of your medicines, including over-the-counter products, supplements and herbal remedies, to every pharmacy visit.

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Domande frequenti

Can I take Propranolol with Thioridazine?

MediHelp rates the interaction as contraindicated. Propranolol and Thioridazine are not normally used together. Taking them at the same time is expected to cause harm or make one of them unsafe, so a different medicine is usually chosen for one of the two. Thioridazine can raise propranolol concentrations, and propranolol can raise thioridazine concentrations. Because thioridazine itself prolongs the QT interval, higher levels increase the risk of torsades de pointes and sudden death.

How serious is the interaction between Propranolol and Thioridazine?

MediHelp rates it contraindicated, on a four-level scale (minor, moderate, major, contraindicated) based on published labels and references. What to do, in brief: Avoid concurrent use. If a beta blocker is needed with thioridazine, select one not dependent on CYP2D6 such as atenolol, though thioridazine alternatives are preferred.

What other medicines interact with Propranolol?

MediHelp also lists interactions of Propranolol with, for example, Acebutolol, Adrenaline-articaine, Albuterol. The full list is on the Propranolol page.

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