Drug reference

chlorpheniramine

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Respiratory (Anti Histamine)

Mechanism of action

Chlorpheniramine competes with histamine for the histamine H1 receptor, reversible competitive inhibitor.

Common side effects

  • Sedation
  • Drowsiness
  • Upset Stomach

Contraindications

  • Documented hypersensitivity Lower respiratory disease, eg, asthma (controversial) Preemies & neonates Nursing women Acute asthma, sleep apnea

Related conditions

Frequently asked questions

What drug class is chlorpheniramine?

chlorpheniramine belongs to: Respiratory.

How does chlorpheniramine work?

Chlorpheniramine competes with histamine for the histamine H1 receptor, reversible competitive inhibitor.

What are the common side effects of chlorpheniramine?

Sedation, Drowsiness, Upset Stomach

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