Drug reference

metaxalone

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Musculoskeletal (Muscle Relaxants)

Mechanism of action

General CNS depression; no direct effect on skeletal muscle; may disrupt the spasm-pain-spasm cycle; does not have direct effect on skeletal muscle.

Common side effects

  • Drug-induced gastrointestinal disturbance
  • Dizziness
  • Vomiting
  • Somnolence
  • Headache
  • Nausea

Contraindications

  • Hypersensitivity History of drug-induced hemolytic anemia Significant renal/hepatic impairment

Related conditions

Frequently asked questions

What drug class is metaxalone?

metaxalone belongs to: Musculoskeletal.

How does metaxalone work?

General CNS depression; no direct effect on skeletal muscle; may disrupt the spasm-pain-spasm cycle; does not have direct effect on skeletal muscle.

What are the common side effects of metaxalone?

Drug-induced gastrointestinal disturbance, Dizziness, Vomiting, Somnolence, Headache, Nausea

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