Drug reference

salmeterol

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Respiratory (B2-Agonist)

Mechanism of action

Long-acting beta-2 agonist; action on beta-2 receptors relaxes bronchial smooth muscle with little effect on heart rate, 50 times more selective than albuterol.

Common side effects

  • Headache
  • joint or muscle pain
  • Nasal Congestion

Contraindications

  • Hypersensitivity Asthma treatment without an inhaled corticosteroid

Known interactions (1)

Related conditions

Frequently asked questions

What drug class is salmeterol?

salmeterol belongs to: Respiratory.

How does salmeterol work?

Long-acting beta-2 agonist; action on beta-2 receptors relaxes bronchial smooth muscle with little effect on heart rate, 50 times more selective than albuterol.

What are the common side effects of salmeterol?

Headache, joint or muscle pain, Nasal Congestion

Which drugs interact with salmeterol?

isocarboxazid

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