Referência de medicamentos
Scopolamine
Scopolamine is a medicine in the class respiratory. It is used for irritable bowel syndrome.
- Classe do medicamento: Respiratory
- Indicado para: irritable bowel syndrome
Última atualização
Para profissionais de saúde — apenas referência. Esta página é um resumo breve, não é aconselhamento médico nem substitui a bula oficial ou o julgamento clínico. Verifique sempre antes de prescrever ou dispensar.
O conteúdo clínico desta página está disponível apenas em inglês.
Pontos-chave
- Classe do medicamento
- Respiratory
- Formas farmacêuticas comuns
- adesivo, comprimido
- Concentrações comuns
- 10 mg, 5 mg/5 ml, 1 mg
- Interações conhecidas
- 143 (Grave: 17 · Moderada: 105 · Leve: 21)
- Nomes comerciais
- 19
- Países e mercados
- 3
Para que é usado
Como funciona
Its anticholinergic action exerts a smooth-muscle relaxing/spasmolytic effect. Blockade of the muscarinic receptors in the GI tract is the basis for its use in the treatment of abdominal pain secondary to cramping. Hyoscine butylbromide also binds to nicotinic receptors, which induces a ganglion-blocking effect.
Dose habitual em adultos (resumo da bula)
Nausea & Vomiting (Treatment): 0.3-0.65 mg IV/IM/SC; repeat q6-8hr if necessary
Gravidez e amamentação
- Gravidez
- Unknown Covers hyoscine butylbromide (Buscopan, poorly absorbed by mouth) and hyoscine hydrobromide (patch, tablets). US patch label: no rise in birth defects in observational data; avoid in severe pre-eclampsia (seizures after injection). UK Buscopan: not recommended in pregnancy as a precaution.
- Amamentação
- Safe Hyoscine passes into milk. LactMed: a single dose is unlikely to affect breastfeeding, but long-term use may reduce milk supply or let-down; watch for poor feeding and weight gain. UK Buscopan: not recommended while breastfeeding (no data).
Efeitos adversos relatados
- Drowsiness
- Dry mouth
- Blurred vision
- Dizziness
- Disorientation
Contraindicações
- Hypersensitivity to scopolamine, belladonna alkaloids, or any component in formulation
- Closed-angle glaucoma
Quem deve ter cuidado
- Use caution in patients with benign prostatic hyperplasia, history of seizures or psychosis, ulcerative colitis, hypertension, hyperthyroidism.
- Scopolamine tablets have been discontinued, but Hyoscine N-Butylbromide is still in market.
- May cause CNS depression; caution when operating heavy machinery or tasks which require mental alertness
Informe ao farmacêutico ou ao médico sobre gravidez ou amamentação, doença renal ou hepática, alergias e todos os outros medicamentos ou suplementos que você usa.
Principais interações (143)
- Benzhydrocodone / acetaminophen + Scopolamine Major
- Buprenorphine long-acting + Scopolamine Major
- Buprenorphine subdermal implant + Scopolamine Major
- Buprenorphine transdermal + Scopolamine Major
- Clozapine + Scopolamine Major
- Fentanyl + Scopolamine Major
- Fentanyl intranasal + Scopolamine Major
- Fentanyl iontophoretic transdermal system + Scopolamine Major
- Fentanyl transdermal + Scopolamine Major
- Fentanyl transmucosal + Scopolamine Major
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Outros medicamentos desta classe
Perguntas frequentes
What is Scopolamine used for?
Scopolamine is a medicine in the class respiratory. It is used for Irritable bowel syndrome, Motion sickness, Nausea & vomiting.
What side effects have been reported with Scopolamine?
Drowsiness, Dry mouth, Blurred vision, Dizziness, Disorientation.
Can Scopolamine be taken in pregnancy or while breastfeeding?
Pregnancy: Unknown. Covers hyoscine butylbromide (Buscopan, poorly absorbed by mouth) and hyoscine hydrobromide (patch, tablets). US patch label: no rise in birth defects in observational data; avoid in severe pre-eclampsia (seizures after injection). UK Buscopan: not recommended in pregnancy as a precaution. Breastfeeding: Safe. Hyoscine passes into milk. LactMed: a single dose is unlikely to affect breastfeeding, but long-term use may reduce milk supply or let-down; watch for poor feeding and weight gain. UK Buscopan: not recommended while breastfeeding (no data).
What does Scopolamine interact with?
MediHelp lists 143 known interactions for Scopolamine. Major: 17 · Moderate: 105 · Minor: 21. The most serious include Benzhydrocodone / acetaminophen, Buprenorphine long-acting, Buprenorphine subdermal implant.
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