Drug reference

cefazolin

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Anti Bacterial (Cephalosporins)

Mechanism of action

First-generation semisynthetic cephalosporin that binds to 1 or more penicillin-binding proteins, thereby arresting bacterial cell-wall synthesis and inhibiting bacterial replication; has poor capacity to cross blood-brain barrier; primarily active against skin flora, including S aureus

Common side effects

  • Anorexia
  • Fever
  • Increased transaminases
  • Eosinophilia
  • Diarrhea

Related conditions

Frequently asked questions

What drug class is cefazolin?

cefazolin belongs to: Anti Bacterial.

How does cefazolin work?

First-generation semisynthetic cephalosporin that binds to 1 or more penicillin-binding proteins, thereby arresting bacterial cell-wall synthesis and inhibiting bacterial replication; has poor capacity to cross blood-brain barrier; primarily active against skin flora, including S aureus

What are the common side effects of cefazolin?

Anorexia, Fever, Increased transaminases, Eosinophilia, Diarrhea

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