Drug reference

obeticholic acid

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Gastrointestinal Tract (Miscellaneous(GIT))

Mechanism of action

Farnesoid X receptor (FXR) agonist: FXR is a nuclear receptor expressed in the liver, intestine, kidney, and adipose tissue that regulates a wide variety of target genes critically involved in the control of bile acid synthesis and transport, lipid metabolism, and glucose homeostasis

Common side effects

  • Pruritus
  • Fatigue
  • Reduced HDL-C
  • Abdominal pain

Related conditions

Frequently asked questions

What drug class is obeticholic acid?

obeticholic acid belongs to: Gastrointestinal Tract.

How does obeticholic acid work?

Farnesoid X receptor (FXR) agonist: FXR is a nuclear receptor expressed in the liver, intestine, kidney, and adipose tissue that regulates a wide variety of target genes critically involved in the control of bile acid synthesis and transport, lipid metabolism, and glucose homeostasis

What are the common side effects of obeticholic acid?

Pruritus, Fatigue, Reduced HDL-C, Abdominal pain

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