Drug reference

pentazocine

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Musculoskeletal (Opioids)

Mechanism of action

Narcotic agonist-analgesic of kappa opiate receptors and partial agonist of mu opiate receptors; inhibits ascending pain pathways, which causes alteration in response to pain; produces analgesia, respiratory depression, and sedation

Common side effects

  • Constipation
  • Dizziness
  • Headache
  • Dry Mouth

Related conditions

Frequently asked questions

What drug class is pentazocine?

pentazocine belongs to: Musculoskeletal.

How does pentazocine work?

Narcotic agonist-analgesic of kappa opiate receptors and partial agonist of mu opiate receptors; inhibits ascending pain pathways, which causes alteration in response to pain; produces analgesia, respiratory depression, and sedation

What are the common side effects of pentazocine?

Constipation, Dizziness, Headache, Dry Mouth

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