Referência de medicamentos
Bismuth subsalicylate
Bismuth subsalicylate is a medicine in the class gastrointestinal tract. It is used for diarrhea.
- Classe do medicamento: Gastrointestinal Tract
- Indicado para: diarrhea
Última atualização Fontes: US FDA label
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Pontos-chave
- Classe do medicamento
- Gastrointestinal Tract
- Formas farmacêuticas comuns
- comprimido, solução, suspensão oral, cápsula, pó
- Concentrações comuns
- 262 mg, 525 mg/30 ml, 525 mg/15 ml
- Interações conhecidas
- 35 (Grave: 2 · Moderada: 24 · Leve: 9)
- Nomes comerciais
- 133
- Países e mercados
- 2
Para que é usado
Como funciona
Antimicrobial, anti-inflammatory action (bismuth); antisecretory effect (salicylate).
Dose habitual em adultos (resumo da bula)
Diarrhea, Gas, Upset Stomach, Indigestion, Heartburn, Nausea:2 tablets (262 mg/tab) or 30 mL every hour; maximum daily dose: 8 regular-strength doses or 4 extra-strength doses.
Gravidez e amamentação
- Gravidez
- Unsafe The salicylate part is absorbed and acts like aspirin: risk of fetal kidney problems, low amniotic fluid and ductus closure later in pregnancy, and bleeding near term. Avoid in pregnancy; use oral rehydration and, if needed, loperamide.
- Amamentação
- Unsafe No direct data; salicylate may pass to the infant through milk. LactMed prefers alternatives. Avoid; use rehydration or loperamide if needed.
Efeitos adversos relatados
- Diarrhea
- Nausea
- Abdominal pain
- Melena
Contraindicações
- Hypersensitivity to bismuth, aspirin, other salicylates
- Infectious diarrhea, high fever, von Willebrand disease, hemorrhage, ulcer or GI bleeding with black or bloody stool, hemophilia
- In pediatric patients, chicken pox or influenza (risk of Reye syndrome)
Quem deve ter cuidado
- Bismuth subcitrate potassium may cause temporary and harmless darkening of tongue and/or black stools, generally reversible within several days after treatment stopped.
- Bismuth absorbs x-rays and may interfere with x-ray diagnostic procedures of gastrointestinal tract.
- Not to be administered to children or teenagers recovering from flu-like symptoms or chickenpox; increased incidence of Reye syndrome, associated with salicylate products
Informe ao farmacêutico ou ao médico sobre gravidez ou amamentação, doença renal ou hepática, alergias e todos os outros medicamentos ou suplementos que você usa.
Principais interações (35)
- Bismuth subsalicylate + Dichlorphenamide Major
- Bismuth subsalicylate + Warfarin Major
- Acetylsalicylic acid + Bismuth subsalicylate Moderate
- Amlodipine-benazepril + Bismuth subsalicylate Moderate
- Aspirin + Bismuth subsalicylate Moderate
- Aspirin / citric acid / sodium bicarbonate + Bismuth subsalicylate Moderate
- Aspirin rectal + Bismuth subsalicylate Moderate
- Atenolol + Bismuth subsalicylate Moderate
- Benazepril + Bismuth subsalicylate Moderate
- Betaxolol + Bismuth subsalicylate Moderate
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- Dosing by age, kidney and liver function, and further dose lines
- Renal and hepatic dose adjustments
- Paediatric dosing
- Dosing in older adults
- How to give it
- Pharmacokinetics
- Patient counselling points
- Food interactions
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Outros medicamentos desta classe
Perguntas frequentes
What is Bismuth subsalicylate used for?
Bismuth subsalicylate is a medicine in the class gastrointestinal tract. It is used for Diarrhea, Helicobacter pylori bacteria, Indigestion, Traveler's diarrhea.
What side effects have been reported with Bismuth subsalicylate?
Diarrhea, Nausea, Abdominal pain, Melena.
Can Bismuth subsalicylate be taken in pregnancy or while breastfeeding?
Pregnancy: Unsafe. The salicylate part is absorbed and acts like aspirin: risk of fetal kidney problems, low amniotic fluid and ductus closure later in pregnancy, and bleeding near term. Avoid in pregnancy; use oral rehydration and, if needed, loperamide. Breastfeeding: Unsafe. No direct data; salicylate may pass to the infant through milk. LactMed prefers alternatives. Avoid; use rehydration or loperamide if needed.
What does Bismuth subsalicylate interact with?
MediHelp lists 35 known interactions for Bismuth subsalicylate. Major: 2 · Moderate: 24 · Minor: 9. The most serious include Dichlorphenamide, Warfarin, Acetylsalicylic acid.
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