Drug reference
cholestyramine
For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.
Drug class
Cardiovascular (Anti Hyperlipidemics)
Mechanism of action
Forms complex with bile acids that is not absorbed through intestine; inhibits enterohepatic reuptake of intestinal bile salts, and this, in turn, increases fecal loss of bile salt-bound LDL and consequently reduces serum cholesterol in patients with primary hypercholesterolemia
Common side effects
- Flatulence
- Constipation
- Belching
- Dental erosion
- Duodenal ulcer bleeding
- Gallstones
- Diarrhea
Related conditions
Frequently asked questions
What drug class is cholestyramine?
cholestyramine belongs to: Cardiovascular.
How does cholestyramine work?
Forms complex with bile acids that is not absorbed through intestine; inhibits enterohepatic reuptake of intestinal bile salts, and this, in turn, increases fecal loss of bile salt-bound LDL and consequently reduces serum cholesterol in patients with primary hypercholesterolemia
What are the common side effects of cholestyramine?
Flatulence, Constipation, Belching, Dental erosion, Duodenal ulcer bleeding, Gallstones, Diarrhea
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