Drug reference

ezetimibe

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Cardiovascular (Anti Hyperlipidemics)

Mechanism of action

Inhibits sterol transporter at brush border and, consequently, intestinal absorption of cholesterol, which in turn decreases delivery of cholesterol to the liver and reduces hepatic cholesterol stores

Common side effects

  • Arthralgia
  • Cough
  • Upper respiratory tract symptoms
  • Pain in extremity
  • Sinusitis
  • Diarrhea

Related conditions

Frequently asked questions

What drug class is ezetimibe?

ezetimibe belongs to: Cardiovascular.

How does ezetimibe work?

Inhibits sterol transporter at brush border and, consequently, intestinal absorption of cholesterol, which in turn decreases delivery of cholesterol to the liver and reduces hepatic cholesterol stores

What are the common side effects of ezetimibe?

Arthralgia, Cough, Upper respiratory tract symptoms, Pain in extremity, Sinusitis, Diarrhea

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