Drug reference

esmolol

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Cardiovascular (Beta Blockers)

Mechanism of action

Class II antiarrhythmic; selective beta1-blocker with little or no effect on beta2 receptors except at high doses. It does not have intrinsic sympathomimetic activity

Common side effects

  • Injection site pain
  • Agitation
  • Dizziness
  • Somnolence
  • Nausea
  • Hypotension

Contraindications

  • Hypersensitivity Sinus bradycardia, 2°/3° heart block, cardiogenic shock, overt cardiac failure Asthma/COPD Sick sinus syndrome without permanent pacemaker

Related conditions

Frequently asked questions

What drug class is esmolol?

esmolol belongs to: Cardiovascular.

How does esmolol work?

Class II antiarrhythmic; selective beta1-blocker with little or no effect on beta2 receptors except at high doses. It does not have intrinsic sympathomimetic activity

What are the common side effects of esmolol?

Injection site pain, Agitation, Dizziness, Somnolence, Nausea, Hypotension

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