Drug reference

tibolone

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Endocrine (Miscellaneous(Hormones))

Mechanism of action

Tibolone appears to regulate estrogenic activity in the various tissues by influencing the availability of estrogenic compounds for the estradiol receptor in a tissue-selective manner.

Common side effects

  • Lower abdominal pain
  • Vaginal discharge
  • Abnormal hair growth
  • Endometrial was thickening

Related conditions

Frequently asked questions

What drug class is tibolone?

tibolone belongs to: Endocrine.

How does tibolone work?

Tibolone appears to regulate estrogenic activity in the various tissues by influencing the availability of estrogenic compounds for the estradiol receptor in a tissue-selective manner.

What are the common side effects of tibolone?

Lower abdominal pain, Vaginal discharge, Abnormal hair growth, Endometrial was thickening

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