Drug reference
granisetron
For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.
Drug class
Gastrointestinal Tract (5-HT3 Antagonist)
Mechanism of action
Selective 5-HT3 receptor antagonist; granisetron binds to 5-HT3 receptors both in the peripheral and central nervous system with primary effects in GI tract.
Common side effects
- Constipation
- Sedation
- Somnolence
- Headache
- Diarrhea
Contraindications
- Hypersensitivity to drug or excipients
Known interactions (3)
Related conditions
Frequently asked questions
What drug class is granisetron?
granisetron belongs to: Gastrointestinal Tract.
How does granisetron work?
Selective 5-HT3 receptor antagonist; granisetron binds to 5-HT3 receptors both in the peripheral and central nervous system with primary effects in GI tract.
What are the common side effects of granisetron?
Constipation, Sedation, Somnolence, Headache, Diarrhea
Which drugs interact with granisetron?
dronedarone, pimozide, thioridazine
Full monographs, dosing and an interaction checker in the MediHelp app
Open the complete reference, check multi-drug interactions and use dosing tools in the MediHelp app.