医薬品リファレンス
Frovatriptan
Frovatriptan is a medicine in the class central nervous system. It is used for migraine.
- 薬効分類: Central Nervous System
- 効能・効果: migraine
最終更新日
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要点
- 薬効分類
- Central Nervous System
- 一般的な剤形
- 錠剤
- 一般的な規格
- 2.5 mg
- 既知の相互作用
- 129 (併用禁忌: 12 · 重大: 8 · 中等度: 78 · 軽度: 31)
- 商品名
- 1
- 国・市場
- 1
何に使われるか
作用のしくみ
Selective 5-HT1 receptor agonist in cranial arteries Causes vasoconstriction and reduces inflammation associated with antidronic neuronal transmission associated with relief of migraine
成人の通常用量(添付文書の要約)
2.5 mg PO at onset; may repeat after 2 hr if migraine recurs; not to exceed 7.5 mg/day
妊娠と授乳
- 妊娠
- Unknown Human data are very limited; registries for triptans (mainly sumatriptan) show no rise in birth defects. Use only if needed; sumatriptan has the most pregnancy data.
- 授乳
- Unknown No published data. UK label: not recommended unless clearly needed; if used, avoid breastfeeding for 24 hours. Triptans can occasionally cause painful nipples. LactMed: an alternative may be preferred, especially with a newborn.
報告されている副作用
- Headache
- Fatigue
- Dizziness
- Chest pain
- Paresthesia
- Hot or cold sensation
注意が必要な方
- Use in peripheral vascular disease, or ischemic bowel disease, or uncontrolled hypertension is contraindicated
- Serotonin syndrome may occur particularly during co-administration with (SSRIs), (SNRIs), (TCAs), and (MOAIs)
- Life-threatening disturbances of cardiac rhythm including ventricular tachycardia and ventricular fibrillation leading to death reported
妊娠中または授乳中であること、腎臓や肝臓の病気、アレルギー、ほかに使用しているすべての薬やサプリメントについて、薬剤師または医師にお伝えください。
主な相互作用 (129)
- Almotriptan + Frovatriptan Contraindicated
- Dihydroergotamine + Frovatriptan Contraindicated
- Dihydroergotamine intranasal + Frovatriptan Contraindicated
- Eletriptan + Frovatriptan Contraindicated
- Ergoloid mesylates + Frovatriptan Contraindicated
- Ergotamine + Frovatriptan Contraindicated
- Frovatriptan + Methylergonovine Contraindicated
- Frovatriptan + Naratriptan Contraindicated
- Frovatriptan + Rizatriptan Contraindicated
- Frovatriptan + Sumatriptan Contraindicated
Pro+会員向け
ページ全体を見る
アカウントを作成してPro+トライアルを始めると、Frovatriptanの完全なモノグラフ(用量、妊娠・授乳、副作用、警告、すべての相互作用)を表示できます。
- Dosing by age, kidney and liver function, and further dose lines
- Paediatric dosing
- Patient counselling points
- Food interactions
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同じ分類のほかの薬剤
よくある質問
What is Frovatriptan used for?
Frovatriptan is a medicine in the class central nervous system. It is used for Migraine.
What side effects have been reported with Frovatriptan?
Headache, Fatigue, Dizziness, Chest pain, Paresthesia, Hot or cold sensation.
Can Frovatriptan be taken in pregnancy or while breastfeeding?
Pregnancy: Unknown. Human data are very limited; registries for triptans (mainly sumatriptan) show no rise in birth defects. Use only if needed; sumatriptan has the most pregnancy data. Breastfeeding: Unknown. No published data. UK label: not recommended unless clearly needed; if used, avoid breastfeeding for 24 hours. Triptans can occasionally cause painful nipples. LactMed: an alternative may be preferred, especially with a newborn.
What does Frovatriptan interact with?
MediHelp lists 129 known interactions for Frovatriptan. Contraindicated: 12 · Major: 8 · Moderate: 78 · Minor: 31. The most serious include Almotriptan, Dihydroergotamine, Dihydroergotamine intranasal.
完全なモノグラフ、用量、相互作用チェッカーはMediHelpアプリで
MediHelpアプリで、完全なリファレンスを開き、複数薬剤の相互作用をチェックし、用量ツールを利用できます。