Drug reference

brexpiprazole

For healthcare professionals — reference only. This page is a brief summary, not medical advice and not a substitute for official labeling or clinical judgement. Always verify before prescribing or dispensing.

Drug class

Central Nervous System (Anti Psychotic (atypical))

Mechanism of action

Serotonin-dopamine activity modulator (SDAM) that acts as a partial agonist at 5-HT1A and dopamine D2 receptors at similar potency, and an antagonist at 5-HT2A and noradrenaline alpha1B/2C receptors

Common side effects

  • Tremor
  • Nasopharyngitis
  • Somnolence
  • Headache
  • Akathisia
  • Increased weight

Known interactions (1)

Related conditions

Frequently asked questions

What drug class is brexpiprazole?

brexpiprazole belongs to: Central Nervous System.

How does brexpiprazole work?

Serotonin-dopamine activity modulator (SDAM) that acts as a partial agonist at 5-HT1A and dopamine D2 receptors at similar potency, and an antagonist at 5-HT2A and noradrenaline alpha1B/2C receptors

What are the common side effects of brexpiprazole?

Tremor, Nasopharyngitis, Somnolence, Headache, Akathisia, Increased weight

Which drugs interact with brexpiprazole?

amisulpride

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